About N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide
N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide (PubChem CID 122497242) has the molecular formula C22H26ClN5O3
and a molecular weight of 443.94 g/mol. Its IUPAC name is N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide.
Molecular Properties
| Compound Name | N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide |
| PubChem CID | 122497242 |
| Molecular Formula | C22H26ClN5O3 |
| Molecular Weight | 443.94 g/mol |
| Exact Mass | 443.17 |
| IUPAC Name | N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide |
| SMILES | CC(=O)N[C@@H](C)COC1CC(COc2ncnc(NCc3cccc(C#N)c3)c2Cl)C1 |
| InChI | InChI=1S/C22H26ClN5O3/c1-14(28-15(2)29)11-30-19-7-18(8-19)12-31-22-20(23)21(26-13-27-22)25-10-17-5-3-4-16(6-17)9-24/h3-6,13-14,18-19H,7-8,10-12H2,1-2H3,(H,28,29)(H,25,26,27)/t14-,18?,19?/m0/s1 |
| InChIKey | SHKSXFSFAIOKMM-YCMKEVRSSA-N |
| XLogP | 3.31 |
| TPSA | 109.16 Ų |
| H-Bond Donors | 2 |
| H-Bond Acceptors | 7 |
| Rotatable Bonds | 10 |
| Heavy Atoms | 31 |
| Complexity | — |
Lipinski Rule of Five
Passes Rule of Five
| Rule | Value |
| MW ≤ 500 | 443.94 |
| LogP ≤ 5 | 3.31 |
| H-Bond Donors ≤ 5 | 2 |
| H-Bond Acceptors ≤ 10 | 7 |
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Frequently Asked Questions
What is the IUPAC name of N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide?
The IUPAC name of N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide (CID 122497242) is N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide.
What is the SMILES notation for N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide?
The canonical SMILES for N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide is CC(=O)N[C@@H](C)COC1CC(COc2ncnc(NCc3cccc(C#N)c3)c2Cl)C1.
What is the InChIKey of N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide?
The InChIKey is SHKSXFSFAIOKMM-YCMKEVRSSA-N. The full InChI is InChI=1S/C22H26ClN5O3/c1-14(28-15(2)29)11-30-19-7-18(8-19)12-31-22-20(23)21(26-13-27-22)25-10-17-5-3-4-16(6-17)9-24/h3-6,13-14,18-19H,7-8,10-12H2,1-2H3,(H,28,29)(H,25,26,27)/t14-,18?,19?/m0/s1.
What are the key properties of N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide?
N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide has a molecular weight of 443.94 g/mol, XLogP of 3.31, 10 rotatable bonds, 2 hydrogen bond donors, and 7 hydrogen bond acceptors.
Where does this data come from?
All data for N-[(2S)-1-[3-[[5-chloro-6-[(3-cyanophenyl)methylamino]pyrimidin-4-yl]oxymethyl]cyclobutyl]oxypropan-2-yl]acetamide is sourced from PubChem (CID 122497242), the world's largest open chemistry database maintained by the National Library of Medicine (NIH).