About 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide
5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide (PubChem CID 137447781) has the molecular formula C29H31FN6O4
and a molecular weight of 546.60 g/mol. Its IUPAC name is 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide.
Molecular Properties
| Compound Name | 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide |
| PubChem CID | 137447781 |
| Molecular Formula | C29H31FN6O4 |
| Molecular Weight | 546.60 g/mol |
| Exact Mass | 546.24 |
| IUPAC Name | 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide |
| SMILES | CNC(=O)c1ccc(NC(=O)C(Cc2ccn(C)n2)n2cc(OC)c(-c3cc(F)ccc3C(C)C)cc2=O)cn1 |
| InChI | InChI=1S/C29H31FN6O4/c1-17(2)21-8-6-18(30)12-22(21)23-14-27(37)36(16-26(23)40-5)25(13-19-10-11-35(4)34-19)29(39)33-20-7-9-24(32-15-20)28(38)31-3/h6-12,14-17,25H,13H2,1-5H3,(H,31,38)(H,33,39) |
| InChIKey | GSSOKSMXFITZEY-UHFFFAOYSA-N |
| XLogP | 3.70 |
| TPSA | 120.14 Ų |
| H-Bond Donors | 2 |
| H-Bond Acceptors | 8 |
| Rotatable Bonds | 9 |
| Heavy Atoms | 40 |
| Complexity | — |
Lipinski Rule of Five
1 violation
| Rule | Value |
| MW ≤ 500 | 546.60 |
| LogP ≤ 5 | 3.70 |
| H-Bond Donors ≤ 5 | 2 |
| H-Bond Acceptors ≤ 10 | 8 |
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Frequently Asked Questions
What is the IUPAC name of 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide?
The IUPAC name of 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide (CID 137447781) is 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide.
What is the SMILES notation for 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide?
The canonical SMILES for 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide is CNC(=O)c1ccc(NC(=O)C(Cc2ccn(C)n2)n2cc(OC)c(-c3cc(F)ccc3C(C)C)cc2=O)cn1.
What is the InChIKey of 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide?
The InChIKey is GSSOKSMXFITZEY-UHFFFAOYSA-N. The full InChI is InChI=1S/C29H31FN6O4/c1-17(2)21-8-6-18(30)12-22(21)23-14-27(37)36(16-26(23)40-5)25(13-19-10-11-35(4)34-19)29(39)33-20-7-9-24(32-15-20)28(38)31-3/h6-12,14-17,25H,13H2,1-5H3,(H,31,38)(H,33,39).
What are the key properties of 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide?
5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide has a molecular weight of 546.60 g/mol, XLogP of 3.70, 9 rotatable bonds, 2 hydrogen bond donors, and 8 hydrogen bond acceptors.
Where does this data come from?
All data for 5-[[2-[4-(5-fluoro-2-propan-2-ylphenyl)-5-methoxy-2-oxo-1-pyridinyl]-3-(1-methylpyrazol-3-yl)propanoyl]amino]-N-methylpyridine-2-carboxamide is sourced from PubChem (CID 137447781), the world's largest open chemistry database maintained by the National Library of Medicine (NIH).