About 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide
3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide (PubChem CID 153054995) has the molecular formula C22H26ClF2N7O
and a molecular weight of 477.95 g/mol. Its IUPAC name is 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide.
Molecular Properties
| Compound Name | 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide |
| PubChem CID | 153054995 |
| Molecular Formula | C22H26ClF2N7O |
| Molecular Weight | 477.95 g/mol |
| Exact Mass | 477.19 |
| IUPAC Name | 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide |
| SMILES | Cc1cc(NC(=O)c2ncc(Cl)nc2N2CCC3(CC2)CC3)nc(N2CCC(F)(F)CC2)n1 |
| InChI | InChI=1S/C22H26ClF2N7O/c1-14-12-16(30-20(27-14)32-10-6-22(24,25)7-11-32)29-19(33)17-18(28-15(23)13-26-17)31-8-4-21(2-3-21)5-9-31/h12-13H,2-11H2,1H3,(H,27,29,30,33) |
| InChIKey | VIHPFOUHMUUUAG-UHFFFAOYSA-N |
| XLogP | 4.10 |
| TPSA | 87.14 Ų |
| H-Bond Donors | 1 |
| H-Bond Acceptors | 7 |
| Rotatable Bonds | 4 |
| Heavy Atoms | 33 |
| Complexity | — |
Lipinski Rule of Five
Passes Rule of Five
| Rule | Value |
| MW ≤ 500 | 477.95 |
| LogP ≤ 5 | 4.10 |
| H-Bond Donors ≤ 5 | 1 |
| H-Bond Acceptors ≤ 10 | 7 |
Analyze 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide with MolForge
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Frequently Asked Questions
What is the IUPAC name of 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide?
The IUPAC name of 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide (CID 153054995) is 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide.
What is the SMILES notation for 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide?
The canonical SMILES for 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide is Cc1cc(NC(=O)c2ncc(Cl)nc2N2CCC3(CC2)CC3)nc(N2CCC(F)(F)CC2)n1.
What is the InChIKey of 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide?
The InChIKey is VIHPFOUHMUUUAG-UHFFFAOYSA-N. The full InChI is InChI=1S/C22H26ClF2N7O/c1-14-12-16(30-20(27-14)32-10-6-22(24,25)7-11-32)29-19(33)17-18(28-15(23)13-26-17)31-8-4-21(2-3-21)5-9-31/h12-13H,2-11H2,1H3,(H,27,29,30,33).
What are the key properties of 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide?
3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide has a molecular weight of 477.95 g/mol, XLogP of 4.10, 4 rotatable bonds, 1 hydrogen bond donors, and 7 hydrogen bond acceptors.
Where does this data come from?
All data for 3-(6-azaspiro[2.5]octan-6-yl)-5-chloro-N-[2-(4,4-difluoropiperidin-1-yl)-6-methylpyrimidin-4-yl]pyrazine-2-carboxamide is sourced from PubChem (CID 153054995), the world's largest open chemistry database maintained by the National Library of Medicine (NIH).