C18H22F3N5O4S — CID 155844076
N-[(5-cyclopropylsulfonyl-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-7-yl)methyl]pyridin-2-amine;2,2,2-trifluoroacetic acid (PubChem CID 155844076) has the molecular formula C18H22F3N5O4S and a molecular weight of 461.47 g/mol. Its IUPAC name is N-[(5-cyclopropylsulfonyl-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-7-yl)methyl]pyridin-2-amine;2,2,2-trifluoroacetic acid.
| Compound Name | N-[(5-cyclopropylsulfonyl-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-7-yl)methyl]pyridin-2-amine;2,2,2-trifluoroacetic acid |
|---|---|
| PubChem CID | 155844076 |
| Molecular Formula | C18H22F3N5O4S |
| Molecular Weight | 461.47 g/mol |
| Exact Mass | 461.13 |
| IUPAC Name | N-[(5-cyclopropylsulfonyl-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepin-7-yl)methyl]pyridin-2-amine;2,2,2-trifluoroacetic acid |
| SMILES | O=C(O)C(F)(F)F.O=S(=O)(C1CC1)N1Cc2ccnn2CC(CNc2ccccn2)C1 |
| InChI | InChI=1S/C16H21N5O2S.C2HF3O2/c22-24(23,15-4-5-15)20-10-13(9-18-16-3-1-2-7-17-16)11-21-14(12-20)6-8-19-21;3-2(4,5)1(6)7/h1-3,6-8,13,15H,4-5,9-12H2,(H,17,18);(H,6,7) |
| InChIKey | OWHAXFAEKDOEGK-UHFFFAOYSA-N |
| XLogP | 1.95 |
| TPSA | 117.42 Ų |
| H-Bond Donors | 2 |
| H-Bond Acceptors | 7 |
| Rotatable Bonds | 5 |
| Heavy Atoms | 31 |
| Complexity | — |
Passes Rule of Five
| Rule | Value |
|---|---|
| MW ≤ 500 | 461.47 |
| LogP ≤ 5 | 1.95 |
| H-Bond Donors ≤ 5 | 2 |
| H-Bond Acceptors ≤ 10 | 7 |