About 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one
3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one (PubChem CID 171648222) has the molecular formula C20H24F3N7O2
and a molecular weight of 451.45 g/mol. Its IUPAC name is 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one.
Molecular Properties
| Compound Name | 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one |
| PubChem CID | 171648222 |
| Molecular Formula | C20H24F3N7O2 |
| Molecular Weight | 451.45 g/mol |
| Exact Mass | 451.19 |
| IUPAC Name | 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one |
| SMILES | Cc1cnc(N2CCN(C(=O)CN3CCCC3c3cc(C(F)(F)F)c(=O)[nH]n3)CC2)nc1 |
| InChI | InChI=1S/C20H24F3N7O2/c1-13-10-24-19(25-11-13)29-7-5-28(6-8-29)17(31)12-30-4-2-3-16(30)15-9-14(20(21,22)23)18(32)27-26-15/h9-11,16H,2-8,12H2,1H3,(H,27,32) |
| InChIKey | TURXKNHHTSPWGP-UHFFFAOYSA-N |
| XLogP | 1.37 |
| TPSA | 98.32 Ų |
| H-Bond Donors | 1 |
| H-Bond Acceptors | 7 |
| Rotatable Bonds | 4 |
| Heavy Atoms | 32 |
| Complexity | — |
Lipinski Rule of Five
Passes Rule of Five
| Rule | Value |
| MW ≤ 500 | 451.45 |
| LogP ≤ 5 | 1.37 |
| H-Bond Donors ≤ 5 | 1 |
| H-Bond Acceptors ≤ 10 | 7 |
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Frequently Asked Questions
What is the IUPAC name of 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one?
The IUPAC name of 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one (CID 171648222) is 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one.
What is the SMILES notation for 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one?
The canonical SMILES for 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one is Cc1cnc(N2CCN(C(=O)CN3CCCC3c3cc(C(F)(F)F)c(=O)[nH]n3)CC2)nc1.
What is the InChIKey of 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one?
The InChIKey is TURXKNHHTSPWGP-UHFFFAOYSA-N. The full InChI is InChI=1S/C20H24F3N7O2/c1-13-10-24-19(25-11-13)29-7-5-28(6-8-29)17(31)12-30-4-2-3-16(30)15-9-14(20(21,22)23)18(32)27-26-15/h9-11,16H,2-8,12H2,1H3,(H,27,32).
What are the key properties of 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one?
3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one has a molecular weight of 451.45 g/mol, XLogP of 1.37, 4 rotatable bonds, 1 hydrogen bond donors, and 7 hydrogen bond acceptors.
Where does this data come from?
All data for 3-[1-[2-[4-(5-methylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl]pyrrolidin-2-yl]-5-(trifluoromethyl)-1H-pyridazin-6-one is sourced from PubChem (CID 171648222), the world's largest open chemistry database maintained by the National Library of Medicine (NIH).