About 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea
1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea (PubChem CID 71093649) has the molecular formula C37H31ClF4N8O5
and a molecular weight of 779.15 g/mol. Its IUPAC name is 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea.
Molecular Properties
| Compound Name | 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea |
| PubChem CID | 71093649 |
| Molecular Formula | C37H31ClF4N8O5 |
| Molecular Weight | 779.15 g/mol |
| Exact Mass | 778.20 |
| IUPAC Name | 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea |
| SMILES | N#Cc1ccc(OC(F)F)c(NC(=O)N(c2ccc(C3CNCCO3)cc2Cl)N(C(=O)Nc2ccc(C3CNCCO3)cc2F)c2cc(C#N)ccc2F)c1 |
| InChI | InChI=1S/C37H31ClF4N8O5/c38-25-15-23(33-19-45-9-11-53-33)4-7-30(25)49(37(52)48-29-13-21(17-43)2-8-32(29)55-35(41)42)50(31-14-22(18-44)1-5-26(31)39)36(51)47-28-6-3-24(16-27(28)40)34-20-46-10-12-54-34/h1-8,13-16,33-35,45-46H,9-12,19-20H2,(H,47,51)(H,48,52) |
| InChIKey | XAKYHVJDMSRHLD-UHFFFAOYSA-N |
| XLogP | 6.98 |
| TPSA | 164.01 Ų |
| H-Bond Donors | 4 |
| H-Bond Acceptors | 9 |
| Rotatable Bonds | 8 |
| Heavy Atoms | 55 |
| Complexity | — |
Lipinski Rule of Five
2 violations
| Rule | Value |
| MW ≤ 500 | 779.15 |
| LogP ≤ 5 | 6.98 |
| H-Bond Donors ≤ 5 | 4 |
| H-Bond Acceptors ≤ 10 | 9 |
Computed Properties (RDKit)
| Structural Alerts | {'alert_name': 'Oxygen-nitrogen_single_bond', 'substructure': 'N/A'} |
|---|
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Frequently Asked Questions
What is the IUPAC name of 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea?
The IUPAC name of 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea (CID 71093649) is 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea.
What is the SMILES notation for 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea?
The canonical SMILES for 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea is N#Cc1ccc(OC(F)F)c(NC(=O)N(c2ccc(C3CNCCO3)cc2Cl)N(C(=O)Nc2ccc(C3CNCCO3)cc2F)c2cc(C#N)ccc2F)c1.
What is the InChIKey of 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea?
The InChIKey is XAKYHVJDMSRHLD-UHFFFAOYSA-N. The full InChI is InChI=1S/C37H31ClF4N8O5/c38-25-15-23(33-19-45-9-11-53-33)4-7-30(25)49(37(52)48-29-13-21(17-43)2-8-32(29)55-35(41)42)50(31-14-22(18-44)1-5-26(31)39)36(51)47-28-6-3-24(16-27(28)40)34-20-46-10-12-54-34/h1-8,13-16,33-35,45-46H,9-12,19-20H2,(H,47,51)(H,48,52).
What are the key properties of 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea?
1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea has a molecular weight of 779.15 g/mol, XLogP of 6.98, 8 rotatable bonds, 4 hydrogen bond donors, and 9 hydrogen bond acceptors.
Where does this data come from?
All data for 1-[2-chloro-N-[[5-cyano-2-(difluoromethoxy)phenyl]carbamoyl]-4-morpholin-2-ylanilino]-1-(5-cyano-2-fluorophenyl)-3-(2-fluoro-4-morpholin-2-ylphenyl)urea is sourced from PubChem (CID 71093649), the world's largest open chemistry database maintained by the National Library of Medicine (NIH).