About 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride
4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride (PubChem CID 87620404) has the molecular formula C26H28Cl2N2OS
and a molecular weight of 487.50 g/mol. Its IUPAC name is 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride.
Molecular Properties
| Compound Name | 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride |
| PubChem CID | 87620404 |
| Molecular Formula | C26H28Cl2N2OS |
| Molecular Weight | 487.50 g/mol |
| Exact Mass | 486.13 |
| IUPAC Name | 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride |
| SMILES | C#CCN(c1nc(-c2cc(C)c(OC)cc2Cl)c(C)s1)[C@@H](CC1CC1)c1ccccc1.Cl |
| InChI | InChI=1S/C26H27ClN2OS.ClH/c1-5-13-29(23(15-19-11-12-19)20-9-7-6-8-10-20)26-28-25(18(3)31-26)21-14-17(2)24(30-4)16-22(21)27;/h1,6-10,14,16,19,23H,11-13,15H2,2-4H3;1H/t23-;/m0./s1 |
| InChIKey | NHJNTZDVOJGMLD-BQAIUKQQSA-N |
| XLogP | 7.49 |
| TPSA | 25.36 Ų |
| H-Bond Donors | |
| H-Bond Acceptors | 4 |
| Rotatable Bonds | 8 |
| Heavy Atoms | 32 |
| Complexity | — |
Lipinski Rule of Five
1 violation
| Rule | Value |
| MW ≤ 500 | 487.50 |
| LogP ≤ 5 | 7.49 |
| H-Bond Donors ≤ 5 | 0 |
| H-Bond Acceptors ≤ 10 | 4 |
Computed Properties (RDKit)
| Structural Alerts | {'alert_name': 'triple_bond', 'substructure': 'N/A'} |
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Frequently Asked Questions
What is the IUPAC name of 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride?
The IUPAC name of 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride (CID 87620404) is 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride.
What is the SMILES notation for 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride?
The canonical SMILES for 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride is C#CCN(c1nc(-c2cc(C)c(OC)cc2Cl)c(C)s1)[C@@H](CC1CC1)c1ccccc1.Cl.
What is the InChIKey of 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride?
The InChIKey is NHJNTZDVOJGMLD-BQAIUKQQSA-N. The full InChI is InChI=1S/C26H27ClN2OS.ClH/c1-5-13-29(23(15-19-11-12-19)20-9-7-6-8-10-20)26-28-25(18(3)31-26)21-14-17(2)24(30-4)16-22(21)27;/h1,6-10,14,16,19,23H,11-13,15H2,2-4H3;1H/t23-;/m0./s1.
What are the key properties of 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride?
4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride has a molecular weight of 487.50 g/mol, XLogP of 7.49, 8 rotatable bonds, 0 hydrogen bond donors, and 4 hydrogen bond acceptors.
Where does this data come from?
All data for 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-phenylethyl]-5-methyl-N-prop-2-ynyl-1,3-thiazol-2-amine;hydrochloride is sourced from PubChem (CID 87620404), the world's largest open chemistry database maintained by the National Library of Medicine (NIH).