Bromazepam

NERVOUS SYSTEM

Key facts

Bromazepam is a drug catalogued in DrugCentral. It was first approved by the YEAR INTRODUCED in 1974. DrugCentral lists 1 molecular target, including GABRA1|GABRG2|GABRB2.

• Molecular targets: GABRA1|GABRG2|GABRB2 (1 listed in DrugCentral).
• ATC code: N05BA08 (Benzodiazepine derivatives).
• Molecular formula: C14H10BrN3O; molecular weight 316.16 g/mol.

Mechanism & targets

Molecular targets (1)

Target	Gene	Action	Activity
GABA-A receptor alpha-1/beta-2/gamma-2	GABRA1|GABRG2|GABRB2	unknown	—

Regulatory approvals (1)

Date	Agency	Marketed as	Applicant	Orphan
1974-01-01	YEAR INTRODUCED	—	—

ATC classification

ATC code	Therapeutic hierarchy
N05BA08	NERVOUS SYSTEM › PSYCHOLEPTICS › ANXIOLYTICS › Benzodiazepine derivatives

Reported adverse-event signals

Strongest FDA FAERS disproportionality signals (log-likelihood ratio). A signal is a statistical association in spontaneous reports, not proof that the drug causes the event.

MedDRA term	LLR
Drug abuse	1736.2
Coma	1690.5
Drug use disorder	1457.1
Poisoning deliberate	1166.4
Toxicity to various agents	899.7
Somnolence	743.7
Sopor	727.3
Intentional overdose	620.7
Substance use disorder	609.6
Suicide attempt	459.2
Miosis	442.6
Mydriasis	435.7

Chemical structure

Full physicochemical, ADMET and 3D-structure analysis of Bromazepam is on its molecule page.

• Molecular formula: C₁₄H₁₀BrN₃O
• Molecular weight: 316.16 g/mol
• CAS number: 1812-30-2
• InChIKey: VMIYHDSEFNYJSL-UHFFFAOYSA-N
• PubChem CID: 2441

BrC1=CC=C2NC(=O)CN=C(C3=CC=CC=N3)C2=C1

Frequently asked questions

Answers are generated from the structured data on this page, not written by hand.

How does Bromazepam work?

Its molecular targets in DrugCentral include GABRA1|GABRG2|GABRB2.

When was Bromazepam first approved?

Bromazepam was first approved by the YEAR INTRODUCED in 1974.

What is the chemical formula of Bromazepam?

Bromazepam has the molecular formula C14H10BrN3O and a molecular weight of 316.16 g/mol.

Sources

• DrugCentral drug card 399 — structure, indications, targets, approvals, pharmacologic classes (CC BY-SA 4.0)
• ChEMBL CHEMBL277062 — compound record and bioactivity
• PubChem CID 2441 — chemical identifiers
• DrugBank DB01558 — drug record
• FDA UNII X015L14V0O — substance identity
• FDA Adverse Event Reporting System (openFDA FAERS) — adverse-event signals, as aggregated by DrugCentral

How this page is built: methodology · editorial policy & corrections.