Piperacetazine

Drug profile

Key facts

Piperacetazine is an ofm drug catalogued in DrugCentral. It was first approved by the FDA in 1969. DrugCentral lists 1 molecular target, including HDAC6.

• Approval status: ofm (first approved 1969 by the FDA).
• Molecular targets: HDAC6 (1 listed in DrugCentral).
• Molecular formula: C24H30N2O2S; molecular weight 410.58 g/mol.

Mechanism & targets

Molecular targets (1)

Target	Gene	Action	Activity
Histone deacetylase 6	HDAC6	unknown	IC50 5.66

Regulatory approvals (1)

Date	Agency	Marketed as	Applicant	Orphan
1969-02-03	FDA	—	—

Chemical structure

Full physicochemical, ADMET and 3D-structure analysis of Piperacetazine is on its molecule page.

• Molecular formula: C₂₄H₃₀N₂O₂S
• Molecular weight: 410.58 g/mol
• CAS number: 3819-00-9
• InChIKey: BTFMCMVEUCGQDX-UHFFFAOYSA-N
• PubChem CID: 19675

CC(=O)C1=CC=C2SC3=CC=CC=C3N(CCCN3CCC(CCO)CC3)C2=C1

Frequently asked questions

Answers are generated from the structured data on this page, not written by hand.

How does Piperacetazine work?

Its molecular targets in DrugCentral include HDAC6.

When was Piperacetazine first approved?

Piperacetazine was first approved by the FDA in 1969.

What is the chemical formula of Piperacetazine?

Piperacetazine has the molecular formula C24H30N2O2S and a molecular weight of 410.58 g/mol.

Sources

• DrugCentral drug card 2186 — structure, indications, targets, approvals, pharmacologic classes (CC BY-SA 4.0)
• ChEMBL CHEMBL1584 — compound record and bioactivity
• PubChem CID 19675 — chemical identifiers
• FDA UNII KL6248WNW4 — substance identity
• DailyMed: FDA labels for Piperacetazine — current prescribing information (label search)
• UniProt Q9UBN7 (HDAC6) — target protein

How this page is built: methodology · editorial policy & corrections.