Vesnarinone

Drug profile

Key facts

Vesnarinone is a drug catalogued in DrugCentral. DrugCentral lists 5 molecular targets, including KCNH2, PDE3B|PDE3A and PDE3A.

• Molecular targets: KCNH2, PDE3B|PDE3A, PDE3A and PDE3B (5 listed in DrugCentral).
• Molecular formula: C22H25N3O4; molecular weight 395.46 g/mol.

Mechanism & targets

Molecular targets (5)

Target	Gene	Action	Activity
Potassium voltage-gated channel subfamily H member 2	KCNH2	unknown	IC50 5.96
Phosphodiesterase 3	PDE3B|PDE3A	unknown	IC50 5.21
cGMP-inhibited 3',5'-cyclic phosphodiesterase A	PDE3A	unknown	IC50 4.97
cGMP-inhibited 3',5'-cyclic phosphodiesterase B	PDE3B	unknown	IC50 4.88
Transitional endoplasmic reticulum ATPase	VCP	unknown	—

Chemical structure

Full physicochemical, ADMET and 3D-structure analysis of Vesnarinone is on its molecule page.

• Molecular formula: C₂₂H₂₅N₃O₄
• Molecular weight: 395.46 g/mol
• CAS number: 81840-15-5
• InChIKey: ZVNYJIZDIRKMBF-UHFFFAOYSA-N
• PubChem CID: 5663

COC1=C(OC)C=C(C=C1)C(=O)N1CCN(CC1)C1=CC=C2NC(=O)CCC2=C1

Frequently asked questions

Answers are generated from the structured data on this page, not written by hand.

How does Vesnarinone work?

Its molecular targets in DrugCentral include KCNH2, PDE3B|PDE3A, PDE3A and PDE3B.

What is the chemical formula of Vesnarinone?

Vesnarinone has the molecular formula C22H25N3O4 and a molecular weight of 395.46 g/mol.

Sources

• DrugCentral drug card 2817 — structure, indications, targets, approvals, pharmacologic classes (CC BY-SA 4.0)
• ChEMBL CHEMBL17423 — compound record and bioactivity
• PubChem CID 5663 — chemical identifiers
• DrugBank DB12082 — drug record
• FDA UNII 5COW40EV8M — substance identity
• UniProt Q12809 (KCNH2) — target protein
• UniProt Q14432 (PDE3A) — target protein
• UniProt Q13370 (PDE3B) — target protein
• UniProt P55072 (VCP) — target protein

How this page is built: methodology · editorial policy & corrections.