Olmutinib
ANTINEOPLASTIC AND IMMUNOMODULATING AGENTS
Also known as: BI 1482694, HM 61713, olita, olmutinib HCl, olmutinib hydrochloride
Data last refreshed: (DrugCentral release 2024-11-01)
Key facts
Olmutinib is a drug catalogued in DrugCentral. DrugCentral lists 2 molecular targets, including BTK and EGFR. Recorded indications include Non-small cell lung cancer.
- Molecular targets: BTK and EGFR (2 listed in DrugCentral).
- Indications: Non-small cell lung cancer.
- ATC code: L01EB06 (Epidermal growth factor receptor (EGFR) tyrosine kinase inhibitors).
- Molecular formula: C26H26N6O2S; molecular weight 486.59 g/mol.
Indications & contraindications
Drug–disease relationships curated by DrugCentral (OMOP / SNOMED concepts).
Indications (1)
- Non-small cell lung cancer
Mechanism & targets
Molecular targets (2)
| Target | Gene | Action | Activity |
|---|---|---|---|
| Tyrosine-protein kinase BTK | BTK | unknown | IC50 9.00 |
| Epidermal growth factor receptor | EGFR | inhibitor | IC50 8.04 |
Regulatory approvals (1)
| Date | Agency | Marketed as | Applicant | Orphan |
|---|---|---|---|---|
| — | Korean Food and Drug Administration (KFDA) | — | — |
ATC classification
| ATC code | Therapeutic hierarchy |
|---|---|
L01EB06 | ANTINEOPLASTIC AND IMMUNOMODULATING AGENTS › ANTINEOPLASTIC AGENTS › PROTEIN KINASE INHIBITORS › Epidermal growth factor receptor (EGFR) tyrosine kinase inhibitors |
Chemical structure
Full physicochemical, ADMET and 3D-structure analysis of Olmutinib is on its molecule page.
| Molecular formula | C26H26N6O2S |
|---|---|
| Molecular weight | 486.59 g/mol |
| CAS number | 1353550-13-6 |
| InChIKey | FDMQDKQUTRLUBU-UHFFFAOYSA-N |
| PubChem CID | 54758501 |
Frequently asked questions
Answers are generated from the structured data on this page, not written by hand.
What is Olmutinib used for?
DrugCentral lists the following indications for Olmutinib: Non-small cell lung cancer.
How does Olmutinib work?
Its molecular targets in DrugCentral include BTK and EGFR (inhibitor).
What is the chemical formula of Olmutinib?
Olmutinib has the molecular formula C26H26N6O2S and a molecular weight of 486.59 g/mol.
Browse: all drugs starting with O · drug guides by category · protein targets A–Z.
Sources
- DrugCentral drug card 5210 — structure, indications, targets, approvals, pharmacologic classes (CC BY-SA 4.0)
- ChEMBL CHEMBL3786343 — compound record and bioactivity
- PubChem CID 54758501 — chemical identifiers
- DrugBank DB13164 — drug record
- FDA UNII CHL9B67L95 — substance identity
- UniProt Q06187 (BTK) — target protein
- UniProt P00533 (EGFR) — target protein
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