About 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide
4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide (PubChem CID 58829098) has the molecular formula C35H37F3N6O2
and a molecular weight of 630.70 g/mol. Its IUPAC name is 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide.
Molecular Properties
| Compound Name | 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide |
| PubChem CID | 58829098 |
| Molecular Formula | C35H37F3N6O2 |
| Molecular Weight | 630.70 g/mol |
| Exact Mass | 630.29 |
| IUPAC Name | 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide |
| SMILES | CC1=C(C=C(C=C1)C(=O)NC2=C(C=CC(=C2)C(F)(F)F)C(=O)N3CCCC3)C4=CC5=CN=C(N=C5C=C4)NCCN6CCCCC6 |
| InChI | InChI=1S/C35H37F3N6O2/c1-23-7-8-25(32(45)41-31-21-27(35(36,37)38)10-11-28(31)33(46)44-16-5-6-17-44)20-29(23)24-9-12-30-26(19-24)22-40-34(42-30)39-13-18-43-14-3-2-4-15-43/h7-12,19-22H,2-6,13-18H2,1H3,(H,41,45)(H,39,40,42) |
| InChIKey | GVLUMNCQENIQPI-UHFFFAOYSA-N |
| XLogP | 7.00 |
| TPSA | 90.50 Ų |
| H-Bond Donors | 2 |
| H-Bond Acceptors | 9 |
| Rotatable Bonds | 8 |
| Heavy Atoms | 46 |
| Complexity | 1020 |
Lipinski Rule of Five
2 violations
| Rule | Value |
| MW ≤ 500 | 630.70 |
| LogP ≤ 5 | 7.00 |
| H-Bond Donors ≤ 5 | 2 |
| H-Bond Acceptors ≤ 10 | 9 |
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Frequently Asked Questions
What is the IUPAC name of 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide?
The IUPAC name of 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide (CID 58829098) is 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide.
What is the SMILES notation for 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide?
The canonical SMILES for 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide is CC1=C(C=C(C=C1)C(=O)NC2=C(C=CC(=C2)C(F)(F)F)C(=O)N3CCCC3)C4=CC5=CN=C(N=C5C=C4)NCCN6CCCCC6.
What is the InChIKey of 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide?
The InChIKey is GVLUMNCQENIQPI-UHFFFAOYSA-N. The full InChI is InChI=1S/C35H37F3N6O2/c1-23-7-8-25(32(45)41-31-21-27(35(36,37)38)10-11-28(31)33(46)44-16-5-6-17-44)20-29(23)24-9-12-30-26(19-24)22-40-34(42-30)39-13-18-43-14-3-2-4-15-43/h7-12,19-22H,2-6,13-18H2,1H3,(H,41,45)(H,39,40,42).
What are the key properties of 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide?
4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide has a molecular weight of 630.70 g/mol, XLogP of 7.00, 8 rotatable bonds, 2 hydrogen bond donors, and 9 hydrogen bond acceptors.
Where does this data come from?
All data for 4-methyl-3-[2-(2-piperidin-1-ylethylamino)quinazolin-6-yl]-N-[2-(pyrrolidine-1-carbonyl)-5-(trifluoromethyl)phenyl]benzamide is sourced from PubChem (CID 58829098), the world's largest open chemistry database maintained by the National Library of Medicine (NIH).