Pimethixene
RESPIRATORY SYSTEM
Also known as: calmixen, mepithiathene, pimethixene maleate, pimetixene
Data last refreshed: (DrugCentral release 2024-11-01)
Key facts
Pimethixene is a drug catalogued in DrugCentral. DrugCentral lists 3 molecular targets, including Htr2a, SETD7 and luxR.
- Molecular targets: Htr2a, SETD7 and luxR (3 listed in DrugCentral).
- ATC code: R06AX23 (Other antihistamines for systemic use).
- Molecular formula: C19H19NS; molecular weight 293.43 g/mol.
Mechanism & targets
Molecular targets (3)
| Target | Gene | Action | Activity |
|---|---|---|---|
| 5-hydroxytryptamine receptor 2A | Htr2a | unknown | Ki 8.60 |
| Histone-lysine N-methyltransferase SETD7 | SETD7 | unknown | IC50 5.37 |
| Transcriptional activator protein luxR | luxR | unknown | IC50 4.25 |
ATC classification
| ATC code | Therapeutic hierarchy |
|---|---|
R06AX23 | RESPIRATORY SYSTEM › ANTIHISTAMINES FOR SYSTEMIC USE › ANTIHISTAMINES FOR SYSTEMIC USE › Other antihistamines for systemic use |
Chemical structure
Full physicochemical, ADMET and 3D-structure analysis of Pimethixene is on its molecule page.
| Molecular formula | C19H19NS |
|---|---|
| Molecular weight | 293.43 g/mol |
| CAS number | 314-03-4 |
| InChIKey | NZLVRVYNQYGMAB-UHFFFAOYSA-N |
| PubChem CID | 4822 |
Frequently asked questions
Answers are generated from the structured data on this page, not written by hand.
How does Pimethixene work?
Its molecular targets in DrugCentral include Htr2a, SETD7 and luxR.
What is the chemical formula of Pimethixene?
Pimethixene has the molecular formula C19H19NS and a molecular weight of 293.43 g/mol.
Browse: all drugs starting with P · drug guides by category · protein targets A–Z.
Sources
- DrugCentral drug card 2169 — structure, indications, targets, approvals, pharmacologic classes (CC BY-SA 4.0)
- ChEMBL CHEMBL1523827 — compound record and bioactivity
- PubChem CID 4822 — chemical identifiers
- DrugBank DB13292 — drug record
- FDA UNII T46J20J26F — substance identity
- UniProt Q8WTS6 (SETD7) — target protein
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