Etoperidone

NERVOUS SYSTEM

Key facts

Etoperidone is a drug catalogued in DrugCentral. DrugCentral lists 4 molecular targets, including HTR1A, SLC6A4 and DRD2.

• Molecular targets: HTR1A, SLC6A4, DRD2 and HRH1 (4 listed in DrugCentral).
• ATC code: N06AB09 (Selective serotonin reuptake inhibitors).
• Molecular formula: C19H28ClN5O; molecular weight 377.92 g/mol.

Mechanism & targets

Molecular targets (4)

Target	Gene	Action	Activity
5-hydroxytryptamine receptor 1A	HTR1A	unknown	Ki 7.07
Sodium-dependent serotonin transporter	SLC6A4	unknown	Ki 6.05
D(2) dopamine receptor	DRD2	unknown	Ki 5.64
Histamine H1 receptor	HRH1	unknown	Ki 5.51

ATC classification

ATC code	Therapeutic hierarchy
N06AB09	NERVOUS SYSTEM › PSYCHOANALEPTICS › ANTIDEPRESSANTS › Selective serotonin reuptake inhibitors

Chemical structure

• Molecular formula: C₁₉H₂₈ClN₅O
• Molecular weight: 377.92 g/mol
• CAS number: —
• InChIKey: IZBNNCFOBMGTQX-UHFFFAOYSA-N
• PubChem CID: 40589

CCN1C(=O)N(CCCN2CCN(CC2)C2=CC(Cl)=CC=C2)N=C1CC

Frequently asked questions

Answers are generated from the structured data on this page, not written by hand.

How does Etoperidone work?

Its molecular targets in DrugCentral include HTR1A, SLC6A4, DRD2 and HRH1.

What is the chemical formula of Etoperidone?

Etoperidone has the molecular formula C19H28ClN5O and a molecular weight of 377.92 g/mol.

Sources

• DrugCentral drug card 1111 — structure, indications, targets, approvals, pharmacologic classes (CC BY-SA 4.0)
• ChEMBL CHEMBL1743259 — compound record and bioactivity
• PubChem CID 40589 — chemical identifiers
• DrugBank DB09194 — drug record
• FDA UNII KAI6MVO39Z — substance identity
• UniProt P08908 (HTR1A) — target protein
• UniProt P31645 (SLC6A4) — target protein
• UniProt P14416 (DRD2) — target protein
• UniProt P35367 (HRH1) — target protein

How this page is built: methodology · editorial policy & corrections.