Picrotin

Drug profile

Key facts

Picrotin is a drug catalogued in DrugCentral. DrugCentral lists 4 molecular targets, including GLRA1, GLRA3 and GLRA2.

• Molecular targets: GLRA1, GLRA3, GLRA2 and GLRB (4 listed in DrugCentral).
• Molecular formula: C15H18O7; molecular weight 310.30 g/mol.

Mechanism & targets

Molecular targets (4)

Target	Gene	Action	Activity
Glycine receptor subunit alpha-1	GLRA1	unknown	IC50 5.28
Glycine receptor subunit alpha-3	GLRA3	unknown	IC50 5.22
Glycine receptor subunit alpha-2	GLRA2	blocker	IC50 4.90
Glycine receptor subunit beta	GLRB	blocker	IC50 4.60

Chemical structure

• Molecular formula: C₁₅H₁₈O₇
• Molecular weight: 310.30 g/mol
• CAS number: 21416-53-5
• InChIKey: RYEFFICCPKWYML-QCGISDTRSA-N
• PubChem CID: 442291

CC(C)(O)[C@@H]1[C@H]2OC(=O)[C@@H]1[C@]1(O)C[C@H]3O[C@]33C(=O)O[C@H]2[C@]13C

Frequently asked questions

Answers are generated from the structured data on this page, not written by hand.

How does Picrotin work?

Its molecular targets in DrugCentral include GLRA1, GLRA3, GLRA2 (blocker) and GLRB (blocker).

What is the chemical formula of Picrotin?

Picrotin has the molecular formula C15H18O7 and a molecular weight of 310.30 g/mol.

Sources

• DrugCentral drug card 2163 — structure, indications, targets, approvals, pharmacologic classes (CC BY-SA 4.0)
• ChEMBL CHEMBL478523 — compound record and bioactivity
• PubChem CID 442291 — chemical identifiers
• FDA UNII U06Z6QD7N2 — substance identity
• UniProt P23415 (GLRA1) — target protein
• UniProt O75311 (GLRA3) — target protein
• UniProt P23416 (GLRA2) — target protein
• UniProt P48167 (GLRB) — target protein

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