Cefsulodin

ANTIINFECTIVES FOR SYSTEMIC USE

Key facts

Cefsulodin is a drug catalogued in DrugCentral. It was first approved by the YEAR INTRODUCED in 1981. DrugCentral lists 7 molecular targets, including GRK2, L3MBTL1 and mrcA.

• Molecular targets: GRK2, L3MBTL1, mrcA and TPT1 (7 listed in DrugCentral).
• ATC code: J01DD03 (Third-generation cephalosporins).
• Molecular formula: C22H20N4O8S2; molecular weight 532.54 g/mol.

Mechanism & targets

Molecular targets (7)

Target	Gene	Action	Activity
Beta-adrenergic receptor kinase 1	GRK2	unknown	EC50 7.15
Lethal(3)malignant brain tumor-like protein 1	L3MBTL1	unknown	IC50 7.01
Penicillin-binding protein 1A	mrcA	unknown	IC50 6.52
tRNA 2'-phosphotransferase	TPT1	unknown	IC50 5.77
Penicillin-binding protein 1B	mrcB	unknown	IC50 5.33
Tyrosine-protein phosphatase non-receptor type 11	PTPN11	unknown	IC50 4.77
Protein-tyrosine phosphatase 1C	PTPN6	unknown	IC50 4.68

Regulatory approvals (1)

Date	Agency	Marketed as	Applicant	Orphan
1981-01-01	YEAR INTRODUCED	—	—

ATC classification

ATC code	Therapeutic hierarchy
J01DD03	ANTIINFECTIVES FOR SYSTEMIC USE › ANTIBACTERIALS FOR SYSTEMIC USE › OTHER BETA-LACTAM ANTIBACTERIALS › Third-generation cephalosporins

Chemical structure

Full physicochemical, ADMET and 3D-structure analysis of Cefsulodin is on its molecule page.

• Molecular formula: C₂₂H₂₀N₄O₈S₂
• Molecular weight: 532.54 g/mol
• CAS number: 62587-73-9
• InChIKey: SYLKGLMBLAAGSC-QLVMHMETSA-N
• PubChem CID: 656575

NC(=O)C1=CC=[N+](CC2=C(N3[C@H](SC2)[C@H](NC(=O)[C@@H](C2=CC=CC=C2)S(O)(=O)=O)C3=O)C([O-])=O)C=C1

Frequently asked questions

Answers are generated from the structured data on this page, not written by hand.

How does Cefsulodin work?

Its molecular targets in DrugCentral include GRK2, L3MBTL1, mrcA and TPT1.

When was Cefsulodin first approved?

Cefsulodin was first approved by the YEAR INTRODUCED in 1981.

What is the chemical formula of Cefsulodin?

Cefsulodin has the molecular formula C22H20N4O8S2 and a molecular weight of 532.54 g/mol.

Sources

• DrugCentral drug card 558 — structure, indications, targets, approvals, pharmacologic classes (CC BY-SA 4.0)
• ChEMBL CHEMBL1590946 — compound record and bioactivity
• PubChem CID 656575 — chemical identifiers
• DrugBank DB13499 — drug record
• FDA UNII OV42LHE42B — substance identity
• UniProt P25098 (GRK2) — target protein
• UniProt Q9Y468 (L3MBTL1) — target protein
• UniProt Q06124 (PTPN11) — target protein
• UniProt P29350 (PTPN6) — target protein

How this page is built: methodology · editorial policy & corrections.