Oxprenolol

CARDIOVASCULAR SYSTEM

Key facts

Oxprenolol is an ofm drug catalogued in DrugCentral. DrugCentral lists 4 molecular targets, including ADRB1, ADRB2 and Htr1a. Recorded indications include Angina pectoris, Anxiety, Hypertensive disorder and Ventricular arrhythmia.

• Approval status: ofm.
• Molecular targets: ADRB1, ADRB2, Htr1a and SLC22A1 (4 listed in DrugCentral).
• Indications: Angina pectoris, Anxiety, Hypertensive disorder and Ventricular arrhythmia.
• ATC code: C07AA02 (Beta blocking agents, non-selective).
• Molecular formula: C15H23NO3; molecular weight 265.35 g/mol.

Indications & contraindications

Drug–disease relationships curated by DrugCentral (OMOP / SNOMED concepts).

Indications (4)

• Angina pectoris
• Anxiety
• Hypertensive disorder
• Ventricular arrhythmia

Mechanism & targets

Molecular targets (4)

Target	Gene	Action	Activity
Beta-1 adrenergic receptor	ADRB1	antagonist	Ki 8.11
Beta-2 adrenergic receptor	ADRB2	antagonist	Ki 8.00
5-hydroxytryptamine receptor 1A	Htr1a	unknown	Ki 7.03
Solute carrier family 22 member 1	SLC22A1	unknown	IC50 4.54

Regulatory approvals (1)

Date	Agency	Marketed as	Applicant	Orphan
—	FDA	—	NOVARTIS

ATC classification

ATC code	Therapeutic hierarchy
C07AA02	CARDIOVASCULAR SYSTEM › BETA BLOCKING AGENTS › BETA BLOCKING AGENTS › Beta blocking agents, non-selective
C07BA02	CARDIOVASCULAR SYSTEM › BETA BLOCKING AGENTS › BETA BLOCKING AGENTS AND THIAZIDES › Beta blocking agents, non-selective, and thiazides
C07CA02	CARDIOVASCULAR SYSTEM › BETA BLOCKING AGENTS › BETA BLOCKING AGENTS AND OTHER DIURETICS › Beta blocking agents, non-selective, and other diuretics

Chemical structure

Full physicochemical, ADMET and 3D-structure analysis of Oxprenolol is on its molecule page.

• Molecular formula: C₁₅H₂₃NO₃
• Molecular weight: 265.35 g/mol
• CAS number: 6452-71-7
• InChIKey: CEMAWMOMDPGJMB-UHFFFAOYSA-N
• PubChem CID: 4631

CC(C)NCC(O)COC1=C(OCC=C)C=CC=C1

Frequently asked questions

Answers are generated from the structured data on this page, not written by hand.

What is Oxprenolol used for?

DrugCentral lists the following indications for Oxprenolol: Angina pectoris, Anxiety, Hypertensive disorder and Ventricular arrhythmia.

How does Oxprenolol work?

Its molecular targets in DrugCentral include ADRB1 (antagonist), ADRB2 (antagonist), Htr1a and SLC22A1.

What is the chemical formula of Oxprenolol?

Oxprenolol has the molecular formula C15H23NO3 and a molecular weight of 265.35 g/mol.

Sources

• DrugCentral drug card 2027 — structure, indications, targets, approvals, pharmacologic classes (CC BY-SA 4.0)
• ChEMBL CHEMBL1200745 — compound record and bioactivity
• PubChem CID 4631 — chemical identifiers
• DrugBank DB01580 — drug record
• FDA UNII 519MXN9YZR — substance identity
• DailyMed: FDA labels for Oxprenolol — current prescribing information (label search)
• UniProt P08588 (ADRB1) — target protein
• UniProt P07550 (ADRB2) — target protein
• UniProt O15245 (SLC22A1) — target protein

How this page is built: methodology · editorial policy & corrections.